阿片樣肽受體
外觀
阿片樣肽受體或阿片類受體、阿片受體(英語:Opioid receptors)是一類以阿片樣肽為配體的G蛋白偶聯受體[1][2][3]。內源性類阿片物質包括強啡肽、腦啡肽、內啡肽、endomorphin和nociceptin。 阿片樣肽受體與生長抑素受體(SSTRs)有約40%的相似性。阿片受體廣泛分佈於大腦,且在脊髓與消化道中也有發現。
參考文獻
[編輯]- ^ Dhawan BN, Cesselin F, Raghubir R, Reisine T, Bradley PB, Portoghese PS, Hamon M. International Union of Pharmacology. XII. Classification of opioid receptors. Pharmacol. Rev. December 1996, 48 (4): 567–92. PMID 8981566.
- ^ Janecka A, Fichna J, Janecki T. Opioid receptors and their ligands. Curr Top Med Chem. 2004, 4 (1): 1–17. PMID 14754373.
- ^ Waldhoer M, Bartlett SE, Whistler JL. Opioid receptors. Annu. Rev. Biochem. 2004, 73: 953–90. PMID 15189164. doi:10.1146/annurev.biochem.73.011303.073940.
外部連結
[編輯]- 醫學主題詞表(MeSH):Opioid+Receptors
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